Kurum Yazarı "Menteşe, Emre" İçin Listeleme
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Study of antıoxidant, antimicrobial and anti-xanthine oxidase activities of some 5,6-dimethyl-2-(substituted)-1h-benzimidazoles and their acylhydrazide derivatives
Baltaş, Nimet; Beriş, Fatih Şaban; Menteşe, Emre (Raman Publ, 2017)In this study, a series of 5,6-dimethy1-2-(4-fluoro/chloro/bromo/methyl/nitrobenzy1)-1Hbenzimidazoles were screened for their bovine milk xanthine oxidase (XO) inhibition, antioxidant and antimicrobial activities. Compounds ... -
Synthesis and anticancer activities of some new coumarin derivatives including the triazole ring and their in silico molecular docking studies
Menteşe, Emre; Güner, Adem; Polatlı, Elifsu; Emirik, Mustafa; Bektaş, Hakan; Kahveci, Bahittin (Wiley-V C H Verlag Gmbh, 2020)The synthesis, docking study, and investigation of the anticancer activities of some coumarin derivatives containing the triazole ring are reported in this study. the newly synthesized compounds were screened for their in ... -
Synthesis and antimicrobial activity of some new triazole bridged benzimidazole substituted phthalonitrile and phthalocyanines
Kantar, Günay Kaya; Menteşe, Emre; Beriş, Fatih Şaban; Şaşmaz, Selami; Kahveci, Bahittin (Editura Acad Romane, 2018)In this study, some new phthalonitriles and metallophthalocyanines (Zn, Ni, Co, and Cu) containing triazole bridged benzimidazole moieties were synthesized starting from 2-(3-methylbenzyl)-1H-benzimidazole Newly synthesized ... -
Synthesis and antioxidant activities of some new triheterocyclic compounds containing benzimidazole, thiophene, and 1,2,4-triazole rings
Menteşe, Emre; Yılmaz, Fatih; Baltaş, Nimet; Bekircan, Olcay; Kahveci, Bahittin (Taylor & Francis Ltd, 2015)Various triheterocyclic compounds containing benzimidazole, thiophene, and 1,2,4-triazole rings (3-6) were synthesized and screened for their antioxidant activities. the structures of the synthesized compounds (2-6) were ... -
Synthesis and antioxidant evaluation of some novel benzimidazole derivatives containing a triazole nucleus
Yılmaz, Fatih; Menteşe, Emre; Baltaş, Nimet (Bentham Science Publ Ltd, 2017)Various benzimidazole compounds containing a triazole nucleus were synthesized and screened for their antioxidant activies. the structures of newly synthesized compounds were characterized by H-1 NMR, C-13 NMR and elemental ... -
Synthesis and antioxidant, antiurease and anti-xanthine oxidase activities of some new benzimidazoles bearing triazole, oxadiazole, thiadiazole and imin function
Karaali, Nesrin; Baltaş, Nimet; Menteşe, Emre (Natl Inst Science Communication & Information Resources-Niscair, 2018)In this study, a series of new 2-(4-nitrobenzyl)-1H-benzimidazole derivatives bearing thiosemicarbazide, triazole, oxadiazole and thiadiazole moieties at the 1st position of benzimidazole ring have been synthesized and ... -
Synthesis and biological evaluation of benzimidazolone bridged triheterocyclic compounds
Menteşe, Emre; Güven, Okan; Çalışkan, Nedime; Baltaş, Nimet (Wiley, 2021)A new series of benzimidazolone bridged triheterocyclic compounds bearing thiosemicarbazide, thiadiazole, triazole, moieties was synthesized and then screened for their in vitro urease, alpha-glucosidase, and acetylcholinesterase ... -
Synthesis and biological evaluation of coumarin-amino acid-benzotriazole conjugates
Menteşe, Emre; Çalışkan, Nedime; Sökmen, Bahar Bilgin; Akyüz, Gülay (Springer, 2024)Objective: It is aimed to synthesize new amino acid-conjugated coumarin-benzotriazole molecules and to investigate their acetylcholinesterase, urease, and lipase inhibition properties. Methods: Urease inhibitory activities ... -
Synthesis and biological evaluation of some 1,3-benzoxazol-2(3H)-one hybrid molecules as potential antioxidant and urease inhibitors
Yılmaz, Fatih; Menteşe, Emre; Sökmen, Bahar Bilgin (Wiley, 2020)A new series of 1,3-benzoxazol-2(3H)-one hybrid compounds, including coumarin, isatin 1,3,4-triazole and 1,3,4-thiadiazole moieties, were synthesized and biologically evaluated for their antioxidant capacities and anti-urease ... -
Synthesis and characterisation of some coumarin-1,2,4-triazol-3-thioether hybrid molecules
Yılmaz, Fatih; Menteşe, Emre (Science Reviews 2000 Ltd, 2017)A new series of N'-{[(4-methyl/phenyl-5-phenyl-4H-1,2,4-triazol-3-yl) thio] acetyl}-2-oxo-2H-chromene-3-carbohydrazides was synthesised via the reaction of 2-[(4-methyl/phenyl-5-phenyl-4H-1,2,4-triazol-3-yl) thio] ... -
Synthesis and characterization of new bistriazole quinazolinediones and their urease inhibition activities
Akyüz, Gülay; Menteşe, Emre (Bentham Science Publications, 2023)A new series of bisthiosemicarbazide and bistriazole molecules bridged quinazolinedione was synthesized and characterized by FT-IR, H-1 and C-13-NMR spectral data. Antiurease activities of all new compounds were tested ... -
Synthesis and characterization of ring-type and branched polymers including polyethylene glycols by "click" chemistry
Öztürk, Temel; Meyvacı, Ergül; Bektaş, Hakan; Menteşe, Emre (Springer International Publishing Ag, 2019)Synthesis of ring-type (or branched) polymers including polyethylene glycols was archived via "click" chemistry of 5,6-diazido-2-benzyl-1H-benzimidazole (Di-N-3) [or triazidoacetohydrazide derivative (Tri-N-3)] and terminally ... -
Synthesis and docking studies of novel benzimidazole derivatives containing thiophene and triazole rings as potential urease inhibitors
Akyüz, Gülay; Emirik, Mustafa; Sökmen, B.B.; Menteşe, Emre (Springer, 2022)Abstract: A new series of 5,6-dichloro-benzimidazoles containing thiophene ring derivatives of thiosemicarbazides and triazoles were designed, synthesized and characterized by spectral methods like as IR, 1H-NMR, 13C-NMR ... -
Synthesis and evaluation of alpha-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
Menteşe, Emre; Karaali, Nesrin; Akyüz, Gülay; Yılmaz, Fatih; Ülker, Serdar; Kahveci, Bahittin (Springer, 2016)A new series of 2-substituted quinazolin-4(3H)-one derivatives including coumarin nucleus has been synthesized and screened for their lipase and a-glucosidase inhibition properties. Among the synthesized compounds, ... -
Synthesis and in vitro urease inhibition of some novel benzimidazole-based hydrazones
Menteşe, Emre; Sökmen, Bahar Bilgin (Wiley, 2019)A novel series of N '-(substituted benzylidene)-2-(5,6-dichloro-2-methyl-1H-benzimidazol-1-yl)acetohydrazides and N '-(1-(substituted phenyl)ethylidene)-2-(5,6-dichloro-2-methyl-1H-benzimidazol-1-yl)acetohydrazides were ... -
Synthesis and kinetics studies of N '-(2-(3,5-disubstituted-4H-1,2,4-triazol-4-yl)acetyl)-6/7/8-substituted-2-oxo-2H-chromen-3-carbohydrazide derivatives as potent antidiabetic agents
Menteşe, Emre; Baltaş, Nimet; Bekircan, Olcay (Wiley-V C H Verlag Gmbh, 2019)A novel series of N '-(2-(3,5-disubstituted-4H-1,2,4-triazol-4-yl)acetyl)-6/7/8-substituted-2-oxo-2H-chromen-3-carbohydrazides were synthesized and studied for their alpha-glucosidase inhibition activity. Most of the ... -
Synthesis and molecular docking study of some 5,6-dichloro-2cyclopropyl-1H-benzimidazole derivatives bearing triazole, oxadiazole, and imine functionalities as potent inhibitors of urease
Menteşe, Emre; Bektaş, Hakan; Sökmen, Bahar Bilgin; Emirik, Mustafa; Çakır, Demet; Kahveci, Bahittin (Pergamon-Elsevier Science Ltd, 2017)A new series of benzimidazole compounds including hydrazinecarbothioamide, 1,2,4-triazole, 1,3,4-oxadiazole and imine function were synthesized starting from 5,6-dichloro-2-cyclopropyl-1H-benzimidazole. All of the benzimidazole ... -
Synthesis and molecular docking study of some novel 2,3-disubstituted quinazolin-4(3H)-one derivatives as potent inhibitors of urease
Akyüz, Gülay; Menteşe, Emre; Emirik, Mustafa; Baltaş, Nimet (Academic Press Inc Elsevier Science, 2018)A new series of 2,3-disubstituted quinazolin-4(3H)-one compounds including oxadiazole and furan rings was synthesized. Their inhibitory activities on urease were assessed in vitro. All newly synthesized compounds exhibited ... -
Synthesis and pancreatic lipase inhibitory activities of some 1,2,4-triazol-5(3)-one derivatives
Özdemir, Yusuf; Bekircan, Olcay; Baltaş, Nimet; Menteşe, Emre (Wiley, 2020)In this study, starting from 4-amino-5-(4-chlorobenzyl)-2,4-dihydro-3H-1,2,4-triazole-3-one (1), the 4-Amino-5-(4-chlorobenzyl)-2-undecyl-2,4-dihydro-3H-1,2,4-triazol-3-one (2) was first synthesized and this compound was ... -
Synthesis and pharmacological activities of some new 2-[1-Heptyl-3-(4-methoxybenzyl)-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl] acetohydrazide derivatives
Bekircan, Olcay; Menteşe, Emre; Ülker, Serdar (Walter de Gruyter Gmbh, 2014)In the present investigation, the key intermediate acetohydrazide derivative 5 was synthesized starting from 3-(4-methoxybenzyl)-4-amino-4,5-dihydro-1,2,4-triazol-5-one (1) by a four-step reaction. Thiosemicarbazides 6a-f ...