Ara
Toplam kayıt 17, listelenen: 11-17
Synthesis and evaluation of alpha-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
(Springer, 2016)
A new series of 2-substituted quinazolin-4(3H)-one derivatives including coumarin nucleus has been synthesized and screened for their lipase and a-glucosidase inhibition properties. Among the synthesized compounds, ...
Design, synthesis, and biological evaluation of coumarin-triazole hybrid molecules as potential antitumor and pancreatic lipase agents
(Wiley-V C H Verlag Gmbh, 2017)
The design, synthesis, and investigation of antitumor and anti-lipase activities of some coumarin-triazole hybrid molecules are reported. the synthesis of these hybrid molecules was performed under microwave irradiation ...
Synthesis, molecular docking and biological evaluation of some benzimidazole derivatives as potent pancreatic lipase inhibitors
(Academic Press Inc Elsevier Science, 2018)
In this study, a new series of benzimidazole and bisbenzimidazole derivatives were prepared via the reaction of iminoester hydrochlorides and o-phenylenediamines and then screened for their lipase inhibition properties. ...
Synthesis of novel triazol compounds containing isatin as potential antibacterial and antifungal agents by microwave and conventional methods
(Sage Publishing, 2011)
Microwave irradiation has been used to accelerate the conversion of isatin (1a) and 5-nitroisatin (1b) into their Schiff bases 3-[5?-aryl(alkyl)- 2?,4?-dihydro-1?,2?,4?-triazol-3?-on- 4?-yl]iminoisatin (3a-g) and ...
An efficient synthesis of some new bisbenzimidazoles via microwave technique
(2014)
2,2’-[1,4 (1,3)-Phenylenedi(methylene)]bis-1 H -benzimidazole derivatives were obtained from the reaction of 1,4- or (1,3)-bisiminoester hydrochloride and o -phenylenediamine derivatives under microwave irradiation. Ester ...
A new green protocol for the synthesis of 2-substituted perimidines from hydrazones under catalyst- and solvent-free conditions
(Bulgarian Academy of Sciences, 2018)
A new green protocol was developed for the synthesis of 2-substituted perimidines. The protocol involves a reaction of ethoxy carbonylhydrazone with 1,8-diaminonaphthalene under solvent- and catalyst-free conditions. Simple ...
Bazı yeni potansiyel biyolojik 4-(Arylidenamino)-2, 4-dihidro-3H- 1,2,4-Triazol-3-one bileşiklerinin mikrodalga- destekli sentezi ve pKa değerlerinin belirlenmesi
(2016)
Bu çalışmada,sekiz yeni bazı potansiyel biyolojik aktif 4-(arilidenamino)-2,4-dihidro-1H-1,2,4-triazol-3-on bileşikleri mikrodalga yöntemi kullanılarak sentezlendi. Bu bileşiklerin yapıları farklı spektroskopik yöntemle ...