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Toplam kayıt 9, listelenen: 1-9
A aonvenient synthesis of Bisbenzimidazoles from iminoester hydrochlorides Via Microwave Technique
(Wiley-Blackwell, 2016)
A simple and practical method has been developed for the synthesis of bisbenzimidazoles. Iminoester hydrochlorides of phenylacetic acids were used as intermediates in this reaction with 3,3'-diaminobenzidine under microwave ...
Synthesis and evaluation of alpha-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
(Springer, 2016)
A new series of 2-substituted quinazolin-4(3H)-one derivatives including coumarin nucleus has been synthesized and screened for their lipase and a-glucosidase inhibition properties. Among the synthesized compounds, ...
Efficient synthesis ofbBenzimidazoles containing 1,2,4-triazol-3-one nucleus using microwave technique
(Springer, 2016)
A series of new compounds containing both benzimidazole and 1,2,4-triazol-3-one rings was synthesized by microwave irradiation of mixtures containing 5-(alkyl/phenyl)-4-(4-carboxyphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-ones ...
Synthesis of new fluorine-containing 1,2,4-triazole-5-on derivatives with their anti-urease, anti-xanthine oxidase and antıoxidant activities
(Editura Acad Romane, 2016)
Acetohydrazide derivatives (3a, b) were obtained starting from 3-(2 or 4-fluorobenzyl)-4-amino-4,5-dihydro-1H-1,2,4-triazole-5-one (la, b) by two steps. Compounds 3a, b were converted to the corresponding methylideneacetohydrazide ...
Acetate bridged dinuclear Cu(II) complexes with ferrocene based benzimidazol ligands: Synthesis, spectroscopy, electrochemistry, DFT calculations and catecholase activity
(Pergamon-Elsevier Science Ltd, 2016)
Two new benzimidazole ligands, 1-[(E)-ferrocenylmethylidenehydrazino]-2-{5,6-dichloro-2-[(o-chloro-phenyl)methyl]-1,3-diaza-1H-inden-1-yl}-1-ethanone (1) and 1-[(E)-ferrocenylmethylidenehydrazino]-2-{2-[p-(trifluoromethy ...
Synthesis and study of antitumor activity of some new 2-(4-methoxybenzyl)-1h-benzimidazole derivatives bearing triazole, oxadiazole and ethanol moiety
(Editura Acad Romane, 2016)
A series of novel 1,2-disubstituted benzimidazole derivatives containing hydrazinecarbothioamide (7a-c), 1,2,4-triazole (8a-c) and 1,3,4-oxadiazole (5) moiety were synthesized starting from 2-(4-methoxybenzyl)-1H-benzimidazole. ...
Determination of biological activities and pka at drug active substance in some bisbenzimidazoles derivatives
(Raman Publ, 2016)
Bisbenzimidazole derivatives have known different structures as drug active substance were evaluated for their biological activities such as antiviral and anti-tumor activities. in addition, acid dissociation constants ...
Experimental and theoretical studies of 4-[(4-methyl-5-phenyl-4h1,2,4-tiıazol-3-yl)sulfanyl]benzene-1,2-dicarbonitrile
(Soc Chemists Technologists Madeconia, 2016)
In this study, 4-[(4-methy1-5-pheny1-4H-1,2,4-triazol-3-yl)sulfanyl]benzene-1,2-dicarbonitrile was synthesized and its molecular structure was characterized by means of FT-IR. and X-ray diffraction methods. the crystal is ...
Ferrocenyl-substituted dinuclear Cu(II) complex: Synthesis, spectroscopy, electrochemistry, DFT calculations and catecholase activity
(Elsevier Science Bv, 2016)
A new ferrocenyl-substituted heterocyclic hydrazide ligand and its Cu(II) complex were prepared. the DFT calculations were performed to determine the electronic and molecular structures of the title compounds. the electronic ...