Ara
Toplam kayıt 7, listelenen: 1-7
Design and microwave-assisted synthesis of a novel Mannich base and conazole derivatives and their biological assessment
(Walter de Gruyter, 2021)
4-Amino-5-methyl-2,4-dihydro-3H-1,2,4-triazol-3-one (1) was converted to the corresponding Schiff base (2) by treatment with salicylaldehyde. 1,2,4-Triazoles were then converted to the corresponding Mannich bases containing ...
Design and microwave-assisted synthesis of a novel Mannich base and conazole derivatives and their biological assessment
(Walter de Gruyter, 2021)
4-Amino-5-methyl-2,4-dihydro-3H-1,2,4-triazol-3-one (1) was converted to the corresponding Schiff base (2) by treatment with salicylaldehyde. 1,2,4-Triazoles were then converted to the corresponding Mannich bases containing ...
Conventional and microwave-assisted synthesis of novel 1,2,4-triazole derivatives containing tryptamine skeleton and evaluation of antimicrobial activity
(Bentham Science Publishing, 2021)
1,2,4-Triazole-3-one (3) obtained from tryptamine was transformed to the corresponding carbox(thio)amides via several steps (6a-d). Their reaction with sodium hydroxide performed the 1,2,4triazole derivatives (7a-d). ...
Conventional and microwave irradiated synthesis, biological activity evaluation of highly substituted indole-triazole hybrids
(Elsevier, 2022)
In the present study, a series of new indole-3-carbaldehyde embedded triazole derivatives have been synthesized. 4-{[(1E)-1H-indol-3-ylmethylidene]amino}-5-methyl-2,4-dihydro-3H-1,2,4-triazol-3-one (2) were converted to ...
Structure-based hybridization, microwave prompted synthesis and biological evaluation of novel 4-(2-fluoro-4-nitrophenyl)morpholine derivatives
(Bentham Science Publ Ltd, 2018)
1,3,4-oxadiazole-2-thiole 6 was obtained from 4-(2-fluoro-4-nitrophenyl)morpholine (2) by the reduction of its nitro group and the sequential treatment of the resulting amine with ethyl bro-moacetate, hydrazine hydrate, ...
Synthesis and characterization of some azole derivatives as potential biological and anticancer agents
(Wiley, 2023)
The treatment of 4-{[(1E)-(2,4-dichlorophenyl)methylene]amino}-5-methyl-2,4-dihydro-3H-1,2,4-triazol-3-one (2) was synthesized from 4-amino-5-methyl-2,4-dihydro-3H-1,2,4-triazol-3-one (1). Then ethyl (4-{[(1E)-(2,4-dichl ...
Synthesis of eperezolid-like molecules and evaluation of their antimicrobial activities
(Springer Link, 2012)
3-Fluoro-4-(4-phenylpiperazin-l-yl)aniline (II) prepared from 3,4-difluoro nitrobenzene was converted to the corresponding Schiff bases (III) and (IV) by treatment with 4-methoxybenzaldehyde and indol-3-carbaldehyde, ...