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Toplam kayıt 5, listelenen: 1-5
Bazı Yeni Potansiyel Biyolojik 4-(Arylidenamino)-2, 4-dihidro-3H- 1,2,4-Triazol-3-one Bileşiklerinin Mikrodalga- destekli Sentezi ve pKa Değerlerinin Belirlenmesi
(2016)
Bu çalışmada,sekiz yeni bazı potansiyel biyolojik aktif 4-(arilidenamino)-2,4-dihidro-1H-1,2,4-triazol-3-on bileşikleri mikrodalga yöntemi kullanılarak sentezlendi. Bu bileşiklerin yapıları farklı spektroskopik yöntemle ...
A aonvenient synthesis of Bisbenzimidazoles from iminoester hydrochlorides Via Microwave Technique
(Wiley-Blackwell, 2016)
A simple and practical method has been developed for the synthesis of bisbenzimidazoles. Iminoester hydrochlorides of phenylacetic acids were used as intermediates in this reaction with 3,3'-diaminobenzidine under microwave ...
Synthesis and evaluation of alpha-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
(Springer, 2016)
A new series of 2-substituted quinazolin-4(3H)-one derivatives including coumarin nucleus has been synthesized and screened for their lipase and a-glucosidase inhibition properties. Among the synthesized compounds, ...
Efficient synthesis ofbBenzimidazoles containing 1,2,4-triazol-3-one nucleus using microwave technique
(Springer, 2016)
A series of new compounds containing both benzimidazole and 1,2,4-triazol-3-one rings was synthesized by microwave irradiation of mixtures containing 5-(alkyl/phenyl)-4-(4-carboxyphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-ones ...
A simple and efficient synthesis of novel inhibitors of alpha-glucosidase based on benzimidazole skeleton and molecular docking studies
(Academic Press Inc Elsevier Science, 2016)
A novel series of benzimidazole derivatives were prepared starting from o-phenylenediamine and 4-nitro-o-phenylenediamine with iminoester hydrochlorides. Acidic proton in benzimidazole was exchanged with ethyl bromoacetate, ...