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Toplam kayıt 8967, listelenen: 7950-7969
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Synthesis and study of antitumor activity of some new 2-(4-methoxybenzyl)-1h-benzimidazole derivatives bearing triazole, oxadiazole and ethanol moiety
(Editura Acad Romane, 2016)A series of novel 1,2-disubstituted benzimidazole derivatives containing hydrazinecarbothioamide (7a-c), 1,2,4-triazole (8a-c) and 1,3,4-oxadiazole (5) moiety were synthesized starting from 2-(4-methoxybenzyl)-1H-benzimidazole. ... -
Synthesis and urease inhibition activities of some new schiff bases benzimidazoles containing thiophene ring
(Springer, 2024)Objective: Schiff bases are significant pharmacophores and show varied biological applications such as antiurease, antidiabetic, antioxidant, antifungal, antibacterial, and anticancer. In this study, new Schiff bases ... -
Synthesis and urease inhibition studies of some new quinazolinones
(Wiley, 2021)In this study, novel quinazolinones were designed, synthesized, characterized by FT-IR, H-1-NMR, C-13-NMR spectral data, and LC-MS. New compounds inhibitory activities on urease were assessed. All of the compounds exhibited ... -
Synthesis and urease inhibition study of some new quinazolinone derivatives bearing triazole, thiadiazole, and piperazine moiety
(Wiley, 2018)A new series of 2,3-disubstituted quinazolin-4(3H)-one derivatives bearing triazole and thiadiazole nucleus has been synthesized and then screened for their urease inhibition properties. All synthesized compounds showed ... -
Synthesis of axinyssa digitata extract directed hybrid nanoflower and investigation of its antimicrobial activity
(IEEE, 2022)First time in this study, the antibacterial effects of sponge extracts and -based cupper hybrid nanoflowers (Cu hNFs) were evaluated. Herein, hybrid nanoflowers (Cu hNFs) were produced by combining sponge extract with Cu2+ ... -
Synthesis of 1,2,4-Triazole derivatives and determination of protonation constant
(2009)A microwave irradiation method has been developed for the synhesis of some 1,2,4-triazole derivatives using environmentally benign solvent ethanol in open vessels. Twelve 1,2,4-triazole derivatives were synthesized in good ... -
Synthesis of 4-Amino-4,5-dihydro-1H-1,2,4-triazole-5-ones and their Isatin-3-imine Derivatives
(MDPI, ST ALBAN-ANLAGE 66, 2005)Iminoester hidroklorürler 1 sentezlenmiştir. Bu bileşikler daha sonra ester etoksikarbonil hidrazonlar 2'ye dönüştürüldü ve bunlardan sırasıyla yeni bir ikame edilmiş 4-amino-4,5-dihidro-lH-1,2,4-triazol-5-onlar, 3 serisi ... -
Synthesis of 5-methyl-2,4-dihydro-3H-1,2,4-triazole-3-one's aryl Schiff base derivatives and investigation of carbonic anhydrase and cholinesterase (AChE, BuChE) inhibitory properties
(Academic Press Inc Elsevier Science, 2019)Carbonic anhydrase enzymes (EC 4.2.1.1, CAs) are metalloenzyme families that catalyze the rapid conversion of H2O and CO2 to HCO3- and H+. CAs are found in different tissues where they participate in various significant ... -
Synthesis of Benzimidazole derivatives containing Schiff base exhibiting antiurease activities
(Sivas Cumhuriyet Üniversitesi, 2021)In this study some novel Schiff bases derivatives of benzimidazole containing thiophene ring were designed and synthesized by using various aldehydes. Seven different aromatic aldehydes with various side groups were used ... -
Synthesis of benzimidazoles containing piperazine ring as potential therapeutic agents against diabetes mellitus and antioxidant activities
(Elsevier, 2024)We synthesized a novel 6-(4-substitue-piperazin-1-yl)-2-aryl-1H-benzimidazole derivatives starting from 5-(4-substitue-piperazin-1-yl)-2-nitroaniline with different aldehydes. A quick "onepot" nitro reductive cyclization ... -
Synthesis of eperezolid-like molecules and evaluation of their antimicrobial activities
(Springer Link, 2012)3-Fluoro-4-(4-phenylpiperazin-l-yl)aniline (II) prepared from 3,4-difluoro nitrobenzene was converted to the corresponding Schiff bases (III) and (IV) by treatment with 4-methoxybenzaldehyde and indol-3-carbaldehyde, ... -
Synthesis of hydroxy benzoin/benzil analogs and investigation of their antioxidant, antimicrobial, enzyme inhibition, and cytotoxic activities
(Scientific Technical Research Council Turkey - TUBİTAK, 2021)In this study, hydroxy benzoin (1-7), benzil (8-14), and benzoin/benzil-O-beta-D-glucosides (15-25) were synthesized to investigate their biological activities. An efficient method for synthesizing hydroxy benzoin compounds ... -
Synthesis of long-term stable gold nanoparticles benefiting from red raspberry (Rubus idaeus), strawberry (Fragaria ananassa), and Blackberry (Rubus fruticosus) extracts-gold Ion complexation and investigation of reaction conditions
(Amer Chemical Soc, 2019)We report synthesis of monodispersed, stable, and colloidal gold nanoparticles (Au NPs) using anthocyanin-riched red raspberry (Rubus idaeus), strawberry (Fragaria ananassa), and blackberry (Rubus fruticosus) extracts as ... -
Synthesis of methyl (E)-2′,4″-thiazachalcones and their N-alkyl derivatives, photochemistry with theoretical calculations and antimicrobial activities
(TUBİTAK, 2009)A series of 9 new (E) -thiazachalcones (1-3), and their N -alkyl substituted derivatives (4-6), and stereoselective dimerization products (7-9) were synthesized, then tested for antimicrobial activity against all test ... -
Synthesis of new carbon material produced from human hair and its evaluation as electrochemical supercapacitor
(Taylor & Francis Inc, 2020)In this study, carbon material similar to graphene structure (GLS) was prepared from graphite and the carbonization of Turkish human hair fibers (HHC) and utilized for the modification of electrode to evaluate the ... -
Synthesis of new coumarin containing benzimidazole derivatives
(Science Reviews 2000 Ltd, 2015)This study describes the synthesis of a new series of benzimidazoles that contain a coumarin moiety. the high yielding synthetic reaction was between hydrazide derivatives of benzimidazoles and 3-(1H-benzotriazol-1-ylcar ... -
Synthesis of new coumarin-C-3 benzimidazole hybrids and their urease inhibition studies
(Bentham Science Publications, 2023)A novel series of coumarin-benzimidazole hybrids were designed, synthesized, and extensively characterized using spectral data, including FT-IR, H-1-NMR, and C-13-NMR. Weatherburn's method was used to test new compounds' ... -
Synthesis of new fluorine-containing 1,2,4-triazole-5-on derivatives with their anti-urease, anti-xanthine oxidase and antıoxidant activities
(Editura Acad Romane, 2016)Acetohydrazide derivatives (3a, b) were obtained starting from 3-(2 or 4-fluorobenzyl)-4-amino-4,5-dihydro-1H-1,2,4-triazole-5-one (la, b) by two steps. Compounds 3a, b were converted to the corresponding methylideneacetohydrazide ... -
Synthesis of new perimidine derivatives from the reaction of 1,8-diaminonapthalene with iminoester hydrochlorides
(Science Reviews 2000 Ltd, 2013)An alternative procedure is described for the synthesis of 2-substituted perimidines involving the reaction of 1,8-diaminonapthalene with iminoester hydrochlorides of substituted phenylacetic acids under microwave irradiation. ... -
Synthesis of nonperipherally tetra-[5-(diethylamino)-2-formylphenoxy] substituted metallophthalocyanines and their electrochemistry
(TUBITAK, 2021)3-[5-(diethylamino)-2-formylphenoxy]phthalonitrile (n-TY-CN), metallophthalocyanines n-TY-Co, n-TY-Cu, and n-TY-Mn bearing [5-(diethylamino)-2-formylphenoxy] groups at nonperipheral positions were prepared for the first ...
