Ara
Toplam kayıt 135, listelenen: 111-120
Synthesis and characterization of new bistriazole quinazolinediones and their urease inhibition activities
(Bentham Science Publications, 2023)
A new series of bisthiosemicarbazide and bistriazole molecules bridged quinazolinedione was synthesized and characterized by FT-IR, H-1 and C-13-NMR spectral data. Antiurease activities of all new compounds were tested ...
Microplastic contamination and risk assessment in table salts: Turkey
(Elsevier, 2023)
In this study, the characterization of microplastics of table salts (n = 36) was determined by FT -IR. Then, individuals' exposure to microplastics from table salt consumption was calculated with a deterministic model, and ...
Regioselective syntheses of 2-oxopyridine carbonitrile derivatives and evaluation for antihyperglycemic and antioxidant potential
(Elsevier, 2023)
A library of 2-oxopyridine carbonitriles 1-34 was synthesized by regioselective nucleophilic substitution reactions. In the first step, a one-pot multicomponent reaction yield pyridone intermediates. The resulting pyridone ...
Staphylococcus aureus bacteriophage 52 endolysin exhibits anti-biofilm and broad antibacterial activity against gram-positive bacteria
(Springer, 2023)
Bacteriophage endolysins have been shown to hold great promise as new antibacterial agents for animal and human health in food preservation. In the present study, endolysin from Staphylococcus aureus subsp. aureus ATCC ...
New pyrimidine-N-β-D-glucosides: synthesis, biological evaluation, and molecular docking investigations
(Scientific Technical Research Council Turkey, TÜBİTAK, 2023)
In this study, syntheses of new pyrimidine-coupled N-beta-glucosides and tetra-O-acetyl derivatives were carried out. All glycoconjugates were investigated in comparison with known chemotherapeutic agents in terms of their ...
Benzimidazolone-piperazine/triazole/thiadiazole/furan/thiophene conjugates: Synthesis, in vitro urease inhibition, and in silico molecular docking studies
(Wiley, 2023)
This study describes the synthesis, in vitro urease inhibition, and molecular docking studies of benzimidazolone derivatives incorporating the piperazine, triazole, thiadiazole, furan, thiophene, and thiosemicarbazide ...
Microplastics in branded milk: Dietary exposure and risk assessment
(Elsevier, 2023)
In this study, 14 packaged milk of various brands sold in the Türkiye market was examined. The microplastics were physically characterised under the microscope. Their vibrational spectra were recorded with the ATF/FT-IR ...
Multicomponent diastereoselective synthesis of tetrahydropyridines as α-amylase and α-glucosidase enzymes inhibitors
(2023)
Background: Researchers seeking new drug candidates to treat diabetes mellitus have been exploring bioactive molecules found in nature, particularly tetrahydropyridines (THPs). Methods: A library of THPs (1–31) were ...
Stereo- and Regio-selective benzo- and Benzohalo-conduritols: Anti-diabetes & anti-tumor activity investigation, kinetic and molecular docking studies
(Elsevier, 2023)
In this study, benzoconduritols, benzohalogenoconduritol, and benzodihalogenoconduritols with conduritol-A and –C structures from oxo-norbornene derivative endo-10 b, exo-11 b cleavaged by Lewis acids (BBr3, BCl3, BF3· ...
Synthesis of some benzimidazole-thiophene hybrids as potential urease and lipase inhibitors
(Springer Link, 2023)
In this study, some benzimidazole-thiophene hybrid compounds containing isatin and salicyl moieties were synthesized and investigated for their urease and lipase inhibition properties. Most of the synthesized compounds ...