Ara
Toplam kayıt 28, listelenen: 1-10
A aonvenient synthesis of Bisbenzimidazoles from iminoester hydrochlorides Via Microwave Technique
(Wiley-Blackwell, 2016)
A simple and practical method has been developed for the synthesis of bisbenzimidazoles. Iminoester hydrochlorides of phenylacetic acids were used as intermediates in this reaction with 3,3'-diaminobenzidine under microwave ...
Synthesis and evaluation of alpha-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
(Springer, 2016)
A new series of 2-substituted quinazolin-4(3H)-one derivatives including coumarin nucleus has been synthesized and screened for their lipase and a-glucosidase inhibition properties. Among the synthesized compounds, ...
Effect of propolis in gastric disorders: inhibition studies on the growth of Helicobacter pylori and production of its urease
(Taylor & Francis Ltd, 2016)
There is considerable interest in alternative approaches to inhibit Helicobacter pylori (H. pylori) and thus treat many stomach diseases. Propolis is a pharmaceutical mixture containing many natural bioactive substances. ...
Inhibition properties of propolis extracts to some clinically important enzymes
(Taylor & Francis Ltd, 2016)
The present study was conducted to envisage inhibition effects of propolis on the crucial enzymes, urease, xanthine oxidase (XO) and acetylcholinesterase (AChE). Some of the antioxidant properties of the propolis samples ...
Efficient synthesis ofbBenzimidazoles containing 1,2,4-triazol-3-one nucleus using microwave technique
(Springer, 2016)
A series of new compounds containing both benzimidazole and 1,2,4-triazol-3-one rings was synthesized by microwave irradiation of mixtures containing 5-(alkyl/phenyl)-4-(4-carboxyphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-ones ...
Novel zinc(II)phthalocyanines bearing azo-containing schiff base: Determination of pKa values, absorption, emission, enzyme inhibition and photochemical properties
(Elsevier Science Bv, 2016)
Azo-containing schiff bases are well known and there are many studies about their various properties in literature. However, phthalocyanines bearing azo-containing schiff bases, their spectral, analytical and biological ...
Three seasonal comprehensive evaluation process of Digitalis trojana Ivan's phenolics
(Elsevier Science Bv, 2016)
Digitalis trojana Ivan, a member of Digitalis genus, has highly bioactive properties due to, efficient phenolics. These compounds have shown to convert into each other in a limited time. Seasonal fluctuations of this plant ...
Molecular docking studies and synthesis of novel bisbenzimidazole derivatives as inhibitors of alpha-glucosidase
(Pergamon-Elsevier Science Ltd, 2016)
A series of bisbenzimidazole derivatives starting from o-phenylenediamine and 4-nitro-o-phenylenediamine were prepared with oxalic acid. Most of the reactions were conducted using both the microwave and conventional methods ...
A simple and efficient synthesis of novel inhibitors of alpha-glucosidase based on benzimidazole skeleton and molecular docking studies
(Academic Press Inc Elsevier Science, 2016)
A novel series of benzimidazole derivatives were prepared starting from o-phenylenediamine and 4-nitro-o-phenylenediamine with iminoester hydrochlorides. Acidic proton in benzimidazole was exchanged with ethyl bromoacetate, ...
Metal-organic frameworks based on copper(I) iodide and pyridine-3,5-dicarboxylic acid: Synthesis, crystal structures and luminescent properties
(Pergamon-Elsevier Science Ltd, 2016)
Two metal -organic frameworks (MOFs) with pyridine-3,5-dicarboxylic acid (H(2)pdc), {[(CuI)-I-I][Cu-II(pdc) (H2O)]center dot 1.5MeCN center dot H2O} (1) and {[Cu(MeCN)(4)]center dot 2[(CuI)-I-I]center dot 2[Cu(2)(II)pdc) ...